The first attempt for the preparation of 2-(tert-butyl)-7-(trimethylsilyl)-3-((trimethylsilyl)oxy)-2,3-dihydro-1H-pyrrolo[3,4-c]pyridine-1-one

Abstract

2-(tert-butyl)-7-(trimethylsilyl)-3-((trimethylsilyl)oxy)-2,3-dihydro-1H-pyrrolo[3,4-c]pyridine-1-ones was synthesized based on a modification of the methodology described by us previously.
The described protocol is simple and does not require the use of expensive and toxic catalysts. The method allows the desired products to be obtained in good yields. Moreover, the procedure is operationally simple and can be considered a more environmentally friendly alternative to conventional catalytic methods.